As you understand from the title of the article, the conversation will go today about trenbolone. “But why many faces?” – some readers will be puzzled … Well, I think it is obvious to everyone that the properties of any drug depend primarily on the active substance, so I meant only the difference in the form of release and ether components, which I will discuss below. And first, let’s talk a little about trenbolone as such.
Trenbolone – a close “relative” of nandrolone, is also a derivative of 19-nor-testosterone, but is fundamentally different from nandrolone in its properties. Trenbolone does not show estrogenic activity and does not aromatize. Common to derivatives of 19-nor-testosterone is the presence of progestogen activity, more moderate in the case of trenbolone. A major difference is that trenbolone is not susceptible to 5-alpha reductase, which significantly increases its potential – nandrolone, under the influence of this enzyme turns into inactive dihydronandrolone (which makes nandrolone almost useless for people with a high content of 5-alpha reductase in the body). Largely due to the non-susceptibility of all sorts of transformations in the body, trenbolone has taken its place in veterinary medicine – it can be successfully applied to all types of mammals. Trenbolone is the clear leader in the time of stabilization of the androgen receptor, it surpasses testosterone 3 times in this, but unlike testosterone, it is not as active in some target cells – the prostate and scalp, which gave reason to seriously consider it as a hormone replacement therapy.
In bodybuilding, trenbolone is mainly used for “drying” and for gaining a dry, high-quality mass. Like testosterone, it can be the only steroid in the cycle due to not only high androgenic and anabolic activity, but also a significant increase in the level of IGF-1 and the ability to activate satellite cells. But the use of his “solo” is hardly a good idea – the progestogenic activity of trenbolone, coupled with a strong suppression of endogenous testosterone, is likely to lead to the so-called “trencane” – a strong suppression of libido.
And now, when the main theoretical part is over, I would like to go on to a brief overview of various trenbolone esters and forms of its release.
Trenbolone acetate ester was never produced by official pharmaceutical companies, but was used exclusively in veterinary medicine. Trebolone acetate is probably the most popular precompetitive steroid – it gives the athlete rigidity and definition due to the inability of trenbolone to aromatize and due to the short ester chain. Currently, there is practically no one underground firm, in the “line” of which he would not be present. According to the results of a number of studies, trenbolone (assuming a low level of estrogen in the body) contributes to the burning of subcutaneous fat, which once again proves its necessity on the “drying” cycle. As such, it is better to combine it with non-aromatizing steroids, especially with stanozolol and drostanolone. “But what about the notorious“ tren-dikom, ”you ask,“ is it possible in the absence of testosterone? ” And, on the other hand, adding testosterone to the cycle can lead to fluid retention in the body … Here comes Proviron, which is actually an oral version of dihydrotestosterone – 50-100 mg of Proviron per day will prevent a decrease in libido and will not cause water retention under skin (dihydrotestosterone does not aromatize). The standard dosage of trenbolone acetate is 50-100 mg per day or every other day. This is one of the main drawbacks of acetate ester – the need to make frequent injections due to the short ester chain, due to which the drug is active only one or two days.
I almost forgot to write about another, exotic or extravagant (I do not know how to characterize it more precisely), the version of trenbolone acetate – oral. Once, due to the not-too-high availability of the injection version, trenbolone acetate tablets were in some demand. Now, the producers of this anachronism can be counted on the fingers. The reason is a very low bioavailability due to non-alkylation of the drug and its destruction during the initial passage of the liver. Any small effect was usually observed from taking 125-150 mg (5-6 tablets of 25 mg) per day, which, coupled with a fairly high price, made the drug not very popular in the bodybuilding community, and the wide distribution of the injection version practically put cross.
Unlike acetate ester, trenbolone hexahydrobenzyl carbonate was produced by the French company Negma for use in humans. The drug was out of production a long time ago, but the underground companies picked up the banner that had fallen – on the black market of steroids a large selection of drugs with this active ingredient.
The main difference from the acetate version is a rather long ethereal “tail” containing 8 carbon atoms.yes – accordingly, more rare injections are required (as a rule, 1-2 injections per week are sufficient). Drugs with a longer ester chain, as a rule, give large gains during weight gain. Trenbolone hexahydrobenzylcarbonate is no exception. The usual dosage is 200-600 mg per week. Trenbolone enanthate. Everything said about hexahydrobenzylcarbonate can also be attributed to enanthate. Well, except that his half-life is somewhat shorter. Unsafe trenbolone Well, here I think everything is clear from the name – trenbolone- “base” is devoid of ether and therefore is metabolized as quickly as possible in the body. The properties and the field of application are similar to trenbolone acetate, but require even more frequent injections – 1-2 times a day. Methyltrienolone (metribolone) I wondered for a while – is it worth talking about this steroid at all? Its accessibility on the steroid market in the post-Soviet space is zero . Whether the producers of the underground are guided by a simple economic calculation based on the conservatism of domestic bodybuilders, who in their mass, like twenty years ago, are focused on “methane” and “deck”, or take care of our health. The last, if someone does not understand – a joke. Below, I will explain what its salt is. Metribolone is an extremely powerful steroid, its anabolic activity is 120-300 times more than methyltestosterone, and androgenic – 60-70 times. In fact, this is the methylated version of trenbolone for oral administration. The drug has never been manufactured industrially, and the only human medicine experiment described by official medicine was conducted by the University of Bonn in 1966. His results were disappointing – after 4 weeks of intake by volunteers in the amount of only 1 mg (!) Per day, the danger of irreversible damage to the liver was revealed. High hepatotoxicity put an end to the prospects for the use of the drug in official medicine. What did not prevent a number of underground firms, completely deprived of social responsibility, to organize its production. Stand alone here (do not count for advertising, I just can not fail to mention) the company Hardcorelabs, prone to innovation. They release two drugs containing metribolone in the form of … injections. Of particular interest is the novelty – a drug called Tren-X, containing metribolone and all the trenbolone esters described above. Their percentage is the secret of the company. It is obvious that the introduction of metribolone into the body by injection does not remove the issue of hepatotoxicity from the agenda, but at least the drug lacks the effect of the initial passage of the liver.